Pritchett, Beau P. and Kikuchi, Jun and Numajiri, Yoshitaka and Stoltz, Brian M. (2017) A Fischer Indolization Strategy toward the Total Synthesis of (–)-Goniomitine. Heterocycles, 95 (2). pp. 1245-1253. ISSN 0385-5414. PMCID PMC5502790. doi:10.3987/COM-16-S(S)80. https://resolver.caltech.edu/CaltechAUTHORS:20170706-132827697
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Abstract
A Fischer indolization strategy toward the core of (–)-goniomitine is reported. Initial investigations into the Pd-catalyzed asymmetric allylic alkylation of dihydropyrido[1,2-a]indolone (DHPI) substrates are also discussed.
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Additional Information: | © 2017 The Japan Institute of Heterocyclic Chemistry. Published online: 15th February, 2017. The authors wish to thank NIH-NIGMS (R01GM080269), Amgen, the Gordon and Betty Moore Foundation, and Caltech for financial support. B.P.P. thanks the NSF for a predoctoral fellowship (Grant DGE-1144469). Y. N. thanks Toray Industries Inc. for a postdoctoral fellowship. The authors thank Dr. Scott Virgil (Caltech) and the Caltech Center for Catalysis and Chemical Synthesis, for instrumentation assistance. Katerina Korch is acknowledged for experimental assistance. | ||||||||||||||
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Issue or Number: | 2 | ||||||||||||||
PubMed Central ID: | PMC5502790 | ||||||||||||||
DOI: | 10.3987/COM-16-S(S)80 | ||||||||||||||
Record Number: | CaltechAUTHORS:20170706-132827697 | ||||||||||||||
Persistent URL: | https://resolver.caltech.edu/CaltechAUTHORS:20170706-132827697 | ||||||||||||||
Usage Policy: | No commercial reproduction, distribution, display or performance rights in this work are provided. | ||||||||||||||
ID Code: | 78814 | ||||||||||||||
Collection: | CaltechAUTHORS | ||||||||||||||
Deposited By: | Tony Diaz | ||||||||||||||
Deposited On: | 06 Jul 2017 21:17 | ||||||||||||||
Last Modified: | 05 Apr 2022 17:39 |
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